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  • دکتری (1394)

    شیمی - آلی

    دانشگاه صنعتی خواجه نصیرالدین طوسی، تهران، ایران

  • کارشناسی‌ارشد (1371)

    شیمی - شیمی آلی

    دانشگاه شهید بهشتی، تهران، ایران

  • کارشناسی (1368)

    شیمی - محض

    دانشگاه شهید چمران اهواز،

  • آلودگی های شیمیایی در محیط زیست

    متولد سال 1341 در شهر اهواز متاهل و دارای دو فرزند دارای 28 سال سابقه کار با دستگاههای NMR نود، سیصد و پانصد مگاهرتز طی دوره آموزشی NMR در توکیو ژاپن بمدت 15 روز طی دوره آموزشی NMR یک بعدی و دوبعدی در زوریخ سویس بمدت 32 روز کسب عنوان دانشمند برتر جهان اسلام از سوی کمیته علمی سازمان کنفرانس اسلامی (Comstec) در سال 1387 کسب عنوان دانشمند ISI در سال 2013

    ارتباط

    رزومه

    Design, Synthesis, Molecular Docking, and Kinetic Study of 3-Amino-2, 4-Diarylbenzo [4, 5] Imidazo [1, 2-a] Pyrimidines as Novel, Potent Α-Glucosidase Inhibitor

    Fariba Peytam, Ghazaleh Takalloobanafshi, Toktam Saadattalab, Zahra Emamgholipour, Maryam Norouzbahari, Setareh Moghimi, Loghman Firoozpour, Hamid Reza Bijanzadeh, Mohammad Ali Faramarzi, Somayeh Mojtabavi, Parviz Rashidi-Ranjbar, Alireza Foroumadi
    Journal Papers , 2021 January 18, {Pages }

    Abstract

    Design, Synthesis, Molecular Docking, and Kinetic Study of 3-Amino-2, 4-Diarylbenzo [4, 5] Imidazo [1, 2-a] Pyrimidines as Novel, Potent Α-Glucosidase Inhibitor

    23Na‐NMR Data Based Donor Number and Their Correlation with Solvatochromic Parameters in Binary Solvent Mixtures

    Ali Reza Harifi‐Mood, Fereshteh Sharifi, Hamid Reza Bijanzadeh
    Journal PapersChemistrySelect , Volume 6 , Issue 4, 2021 January 27, {Pages 600-608 }

    Abstract

    Donor numbers (DNs) of binary mixtures of acetonitrile with methanol, ethanol, ethylene glycol, 1‐butanol, and tert‐butanol were calculated in the whole range of mole fractions based on 23Na‐NMR chemical shift of sodium perchlorate dissolved in solvent. Data showed positive deviation from hypothetical linear ideal behavior. Solvatochromic parameters including empirical polarity, dipolar/polarizability, hydrogen bond donor, and hydrogen bond acceptor of the solvent mixtures were spectrophotometrically measured in order to investigate the correlations among parameters. The trend of data showed the preferential solvation along with synergistic behavior in some of mixtures. Applying preferential solvation model confirmed the solvent‐so

    Synthesis of N-(Isoquinolin-1-yl)sulfonamides via Ag2O-Catalyzed Tandem Reaction of ortho-Alkynylbenzaldoximes with Benchtop Stabilized Ketenimines

    Sepideh Hayatgheybi, Hormoz Khosravi, Hossein Zahedian Tejeneki, Frank Rominger, Hamid Reza Bijanzadeh, Saeed Balalaie
    Journal PapersOrganic Letters , 2021 April 14, {Pages }

    Abstract

    In this project, a moderately efficient approach to multisubstituted N-(isoquinolin-1-yl)sulfonamide derivatives was illustrated, utilizing ortho-alkynylbenzaldoximes and zwitterionic ketenimine salts in a tandem reaction catalyzed by silver oxide. The oxophilicity of Ag2O, along with its nature as Lewis acid, pave the way for a smooth [3 + 2] cycloaddition between isoquinoline N-oxides and ketenimine species, which is a key step in this reaction. DFT calculation suggests that 1,3-dipolar cycloaddition of nitrone and ketenimine proceeds through a selective stepwise mechanism.

    Synthesis of Spiro[chromene-imidazo[1,2-a]pyridin]-3′-imines via 6-exo-dig Cyclization Reaction

    B Nayebzadeh, K Amiri, H Khosravi, S Mirzaei, F Rominger, D Dar’in, ...
    Journal Papers , , {Pages }

    Abstract

    Domino Decarboxylative Arylation and C–O Selective Bond Formation toward Chromeno[2,3-b]pyridine-2-one Skeletons

    EM Ahadi, AA Kejani, H Khosravi, VF Vavsari, S Balalaie, F Rominger, ...
    Journal Papers , , {Pages }

    Abstract

    Copper(I)‐Catalyzed Intramolecular Cyclization of o‐Propargyloxy Diketopiperazines to Access Diverse Diazabicyclic and Spiro‐Diketopiperazinochromanes

    B Manavi, HZ Tejeneki, F Rominger, M Armaghan, W Frank, ...
    Journal Papers , , {Pages }

    Abstract

    A Domino Approach for the Synthesis of 4-Carboxamide Oxazolines from Azirines

    A Nikbakht, F Mohammadi, MS Mousavi, K Amiri, S Balalaie, F Rominger, ...
    Journal Papers , , {Pages }

    Abstract

    Design, synthesis, molecular docking, and in vitro α-glucosidase inhibitory activities of novel 3-amino-2, 4-diarylbenzo [4, 5] imidazo [1, 2-a] pyrimidines against yeast and …

    F Peytam, G Takalloobanafshi, T Saadattalab, M Norouzbahari, ...
    Journal Papers , , {Pages }

    Abstract

    Structure-activity relationship studies of Longicalcynin A analogues, as anticancer cyclopeptides

    Mohammadreza Gholibeikian, Abdolhamid Bamoniri, Mohammad Hassan HoushdarTehrani, Bi Bi Fatemeh Mirjalili, Hamid Reza Bijanzadeh
    Journal PapersChemico-Biological Interactions , Volume 315 , 2020 January 5, {Pages 108902 }

    Abstract

    Cancer has emerged as the main cause of the highest rate of mortality in the world. Drugs used in cancer, although, show some beneficial effects on cancerous organs, demonstrate side effects on other normal tissues. On the other hand, anticancer peptides, being effective on target tissues, should be safe and less harmful on healthy organs, since peptides have several advantages, i.e., high activity, specificity, affinity, being less immunogenic and not accumulate in the body. In the present work, analogues of Longicalcynin A, a naturally occurring anticancer cyclopeptide, were synthesized and evaluated their cytotoxicity in order to gain information from structure-activity relationships of the such cyclopeptides which may lead to find novel

    Ultrasound-Activated Atom-Economical Approach to the Synthesis of Highly Substituted Pyrrolidin-2-ones through a Four-Component Ugi/5-endo-trig Intramolecular Radical?…

    Atena Nashta Rahimi, Helya Janatian Ghazvini, Saeed Balalaie, Frank Rominger, Hossein Zahedian Tejeneki, Hamid R Bijanzadeh
    Journal PapersSynlett , Volume 31 , Issue 09, 2020 June , {Pages 871-877 }

    Abstract

    An efficient and diversity-oriented access to functionalized pyrrolidin-2-ones through an Ugi reaction of readily available starting materials with a subsequent transformation is described. A two-step reaction sequence of a four-component Ugi reaction and an intramolecular radical-cyclization reaction leads to the chemo- and regioselective formation of a single product with high atom economy and good to high yields. The radicalization of the pseudopeptides generated from the first step by a cavitational mechanism produces the key intermediate for the ultrasound-activated formation of γ-lactams as the final products by β-Michael addition. Among the advantages of this approach are its use of cavitation bubble implosion as an exclusive path

    Corrigendum to" Structure-activity relationship studies of longicalcynin A analogues, as anticancer cyclopeptides"[Chem. Biol. Interact. 315 (2020) 108902, 1-14].

    Mohammadreza Gholibeikian, Abdolhamid Bamoniri, Mohammad Hassan HoushdarTehrani, Fatemeh Mirjalili BB, Hamid Reza Bijanzadeh
    Journal PapersChemico-Biological Interactions , 2020 June 15, {Pages 109143-109143 }

    Abstract

    Europe PMC is an archive of life sciences journal literature.

    Design, synthesis, molecular docking study, and antibacterial evaluation of some new fluoroquinolone analogues bearing a quinazolinone moiety

    Maryam Norouzbahari, Somayeh Salarinejad, M?mtaz G?ran, Gizem Şanlıt?rk, Zahra Emamgholipour, Hamid Reza Bijanzadeh, Mahsa Toolabi, Alireza Foroumadi
    Journal PapersDARU Journal of Pharmaceutical Sciences , 2020 October 8, {Pages 12-Jan }

    Abstract

    BackgroundIncreasing bacterial resistance to quinolones is concerning. Hence, the development of novel quinolones by chemical modifications to overcome quinolone resistance is an attractive perspective in this context.ObjectiveIn this study, it is aimed to design and synthesize a novel series of functionalized fluoroquinolones using ciprofloxacin and sarafloxacin cores by hybridization of quinazolinone derivatives. This objective was tested by a comprehensive set of in vitro antibacterial assays in addition to SAR (structure–activity relationship) characterisation studies.MethodsA nucleophilic reaction of ciprofloxacin and sarafloxacin with 2-(chloromethyl) quinazolin-4 (3H)-one in the presence of NaHCO 3 in dimethylformamide (DMF) was pe

    Quinazolin-4 (3H)-one based agents bearing thiadiazole-urea: Synthesis and evaluation of anti-proliferative and antiangiogenic activity

    Aram Faraji, Rasoul Motahari, Zaman Hasanvand, Tayebeh Oghabi Bakhshaiesh, Mahsa Toolabi, Setareh Moghimi, Loghman Firoozpour, Mohammad Amin Boshagh, Roya Rahmani, Shima HME Ketabforoosh, Hamid Reza Bijanzadeh, Rezvan Esmaeili, Alireza Foroumadi
    Journal PapersBioorganic Chemistry , 2020 December 13, {Pages 104553 }

    Abstract

    Abstract A series of quinazolin-4 (3H)-one based agents containing thiadiazole-urea were designed, synthesized, and biologically evaluated. The proliferation rate of PC3 cells was moderately reduced by compound 9f (IC 50= 17.7 μ M) which was comparable with sorafenib (IC 50= 17.3 μ M). There was also a significant reduction in the number of HUVEC cells, when they were exposed to compound 9y (IC 50= 6.1 μ M). To test the potential of compounds in inducing apoptosis, Annexin V-FITC/propidium iodide double staining assay was used. After the treatment of HUVEC cells with 9f, they underwent apoptotic effects. A substantial effort was dedicated to gathering comprehensive data across CAM assay. These data showed that 9f moderately inhibits the

    Structure-activity relationship studies of longicalcynin A analogues, as anticancer cyclopeptides (vol 315, 108902, 2020)

    Mohammadreza Gholibeikian, Abdolhamid Bamoniri, Mohammad Hassan HoushdarTehrani, Bi Bi Fatemeh Mirjalili, Hamid Reza Bijanzadeh
    Journal PapersCHEMICO-BIOLOGICAL INTERACTIONS , Volume 331 , 2020 November 1, {Pages }

    Abstract

    Synthesis of Novel Peptides Using Unusual Amino Acids

    Bahareh Talaei, Vaezeh Fathi Vavsari, Saeed Balalaie, Armin Arabanian, Hamid Reza Bijanzadeh
    Journal PapersIranian Journal of Pharmaceutical Research , Volume 19 , Issue 3, 2020 September 1, {Pages 370-382 }

    Abstract

    Small peptides are valuable peptides due to their extended biological activities. Their activities could be categorized according to their low antigenicity, osmotic pressure, and also because of their astonishing bioactivities. For example, the aggression of Phe-Phe fibers via self-assembly and intermolecular hydrogen bonding is the main reason for the formation of Alzheimer’s β-amyloid fibrils. Hydrogen bonding is the main intramolecular interaction in peptides, while the presence of aromatic ring leads to the π-π stacking and affects the self-assembly and aggression. Thus, insertion of an unusual amino acid into peptide sequence facilitates the formation of intramolecular bonds, lipophilicity and its conformation. To design new small

    Ultrasound-Activated Atom-Economical Approach to the Synthesis of Highly Substituted Pyrrolidin-2-ones through a Four-Component Ugi/5-endo-trig Intramolecular Radical …

    AN Rahimi, HJ Ghazvini, S Balalaie, F Rominger, HZ Tejeneki, ...
    Journal Papers , , {Pages }

    Abstract

    Design and Synthesis of Novel Functionalized Fused Oxazepine and Diazepine Analogues Containing Coumarin Backbone through Domino Reaction

    Samane Poursan, Somayeh Ahadi, Saeed Balalaie, Frank Rominger, Hamid Reza Bijanzadeh
    Journal PapersChemistrySelect , Volume 4 , Issue 20, 2019 May 31, {Pages 6403-6407 }

    Abstract

    A simple and straightforward approach has been developed for the synthesis of functionalized fused oxazepine and diazepine analogues containing coumarin backbone. The approach was done through three‐component reaction of 4‐chloro‐3‐formylcoumarin, triphenyl‐λ5‐phosphanylidene derivatives and 2‐aminophenol or o‐phenylenediamine derivatives in the presence of cesium carbonate at room temperature. Carrying out the same reaction without base led to 4‐aminoarylcoumarins. Mild reaction conditions and synthesis of fused functionalized heterocyclic backbones are advantages of this approach.

    Choline Chloride/Urea as Mild Media for the Synthesis of the Chromonyl Amidodiester Fragments and Succinimide Derivatives

    Hoda Jamaati, Saeed Balalaie, Maryam Kazemi Miraki, Frank Rominger, Hamid Reza Bijanzadeh
    Journal PapersChemistrySelect , Volume 4 , Issue 31, 2019 August 23, {Pages 9074-9078 }

    Abstract

    A simple, green protocol has been accomplished for the synthesis of amidoesters 5 a‐k in choline chloride/urea (1:2) through multicomponent reaction of 3‐formyl chromone, Meldrum's acid, isocyanides and primary alcohols via a domino reaction. Carrying out the reaction using trifluoroethanol led to succinimide derivatives 6 a‐d. Easy work‐up, selectivity, and good to excellent yields are the advantages of this protocol.

    Correction to: Genetically encoded photochemical covalent crosslinking within the Hcp-1 self-assembling bacterial secretion machinery

    Alicja K Antonczak, Kedric Milholland, Eric M Tippmann, Michael P Whyte, Stephen P Coburn, Lawrence M Ryan, Fan Zhang, Vincent Maloney, Zach Szczepanski, Keith Smith, Nataliya Samoylova, Steven Stevenson, Younis Hazari, Arif Bashir, Mudasir Habib, Khalid
    Journal PapersAmino acids , Volume 51 , Issue 3, 2019 March 7, {Pages 577 }

    Abstract

    Article: Enhancement of calcium/vitamin D supplement efficacy by administering concomitantly three key nutrients essential to bone collagen matrix for the treatment of osteopenia in middle-aged women: a one-year follow-up

    Synthesis of Functionalized Dihydropyrido [2, 3-d] pyrimidines in Aqueous Medium

    Saeed Balalaie, Hamed Esmaeilabadi, Saber Mehrparvar, Frank Rominger, Fatima Hamdan, Hamid Reza Bijanzadeh
    Journal PapersSynOpen , Volume 2 , Issue 01, 2018 January , {Pages 0001-0005 }

    Abstract

    Synthesis of functionalized 2,3-dihydropyrido[2,3-d]pyrimidin-4(1H)-one from a cascade reaction between 3-formylchromone, malononitrile, diammonium hydrogen phosphate, and aromatic aldehydes in aqueous media is described.

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    دروس نیمسال جاری

    • دكتري
      عناصر كمياب در محيط زيست ( واحد)
      دانشکده منابع طبیعی و علوم دریایی، گروه محيط زيست

    دروس نیمسال قبل

    • كارشناسي ارشد
      شيمي محيط زيست ( واحد)
      دانشکده منابع طبیعی و علوم دریایی، گروه محيط زيست
    • 1400
      پستادست, معصومه
      ارزيابي پسماند غذايي برپايه ي ارزيابي چرخه ي حيات(LCA) براي بيماران در سيستم مراقبت هاي بهداشتي
    • مدیر امور فرهنگی دانشگاه
      داده ای یافت نشد

    مهم

    جدید

      اطلاعیه ای درج نشده است